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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6S0923 | Hypericin | Hypericine,Cyclosan | Apoptosis , Antiviral , Influenza Virus , Tyrosine Kinases , Antibacterial , PKC |
1. Hypericin (Cyclosan) has antineoplastic activity. 2. Hypericin has antibiotic and antiviral activities. 3. Hypericin has antidepressive activity through inhibiting monoamine oxidase enzyme. 4. Hypericin inhibits RANKL... | |||
T36816 | S-trityl-L-Cysteine | STLC | Kinesin |
S-trityl-L-Cysteine is a non-natural amino acid and an inhibitor of Eg5, also known as KSP and Kif11, a mitotic kinesin necessary for mitotic spindle formation. S-trityl-L-Cysteine inhibits the ATPase activity of Eg5 in ... | |||
T9636 | Dalpiciclib | SHR-6390 | CDK |
Dalpiciclib (SHR-6390) is a highly selective, orally bioavailable, and comparable potency inhibitor of CDK4 and CKD6 with IC50s of 12.4 nM and 9.9 nM, respectively. Dalpiciclib exerts potent antitumor activity in esophag... | |||
T0431 | Abexinostat | CRA 24781,PCI24781,PCI-24781,PCI 24781,CRA 024781 | HDAC |
PCI-24781 (Abexinostat (PCI24781)) is a new pan-HDAC inhibitor mainly targeting HDAC1 (Ki: 7 nM), also have moderate inhibitory for HDACs 2, 3, 6, and 10 and greater than 40-fold selectivity against HDAC8. Phase 1/2. | |||
TQ0245 | Sapacitabine | CS682,CYC682 | Nucleoside Antimetabolite/Analog |
Sapacitabine is a nucleoside analog prodrug with antitumor activity. | |||
T10342 | Antitumor agent-2 | Others | |
Antitumor agent-2 has anti-inflammatory and anti-tumor activity and can be used to study cancer. | |||
T67047 | 2-Acetyl-3-ethylpyrazine | Endogenous Metabolite | |
2-Acetyl-3-ethylpyrazine has antitumor activity. | |||
T67785 | ABI-1968 | ||
ABI-1968 has antiviral and antitumor activity. | |||
T72027 | 6-Methyl-3-pyridinecarboxaldehyde | 6-Methoxynicotinaldehyde | |
6-Methyl-3-pyridinecarboxaldehyde (6-Methoxynicotinaldehyde) has partial antitumor activity. | |||
T7611 | ODM-203 | VEGFR , FGFR | |
ODM-203, a Selective Inhibitor of FGFR and VEGFR, Shows Strong Antitumor Activity, and Induces Antitumor Immunity | |||
T3S1457 | Palmaturbine | Palmatrubin,Palmatrubine | Others |
Palmaturbine (Palmatrubine) shows high antitumor activity. | |||
T13799 | NQO1 substrate | NADPH | |
NQO1 substrate is a highly potent NQO1 substrate with potential antitumor activity for leukemia research. | |||
T23151 | Phortress | NSC 710305 | AhR |
Phortress (NSC-710305) is a potent AhR ligand with strong binding affinity, which subsequently triggers the transcription of CYP1A1 and induces antitumor activity. | |||
TN7217 | 4,6-Benzilidine-D-Glucose | ||
4,6-Benzilidine-D-Glucose is a clinical antitumor compound showing antitumor activity in rats with chemically induced hepatocellular carcinoma. | |||
T9998 | MIND4-19 | Sirtuin | |
MIND4-19 is an inhibitor of SIRT2 with antitumor activity. | |||
T6821 | Dp44mT | Apoptosis , Others , Ferroptosis | |
Dp44mT, a effective iron chelator, has selective antitumor activity. | |||
T16913 | Sotirimod | R850,S-30594 | Virus Protease |
Sotirimod(R850) is a novel immunomodulator with antitumor and antiviral activity for the study of actinic keratoses. | |||
T28189 | Nortopixantrone HCl | BBR3438,Nortopixantrone hydrochloride,BBR-3438 | Others |
Nortopixantrone HCl (BBR 3438) is a novel 9-azacyclonopyrazole that shows antitumor activity in a human prostate cancer model. | |||
T16551 | Pladienolide B | Apoptosis | |
Pladienolide B is a potent spliceosome inhibitor, a macrolide isolated from Streptomyces obtusususus Mer-12, which targets the SF3B1 subunit of the spliceosome.Pladienolide B exerts its antitumor effects by inhibiting pr... | |||
T10276L | AKT Kinase Inhibitor HCl | AKT Kinase Inhibitor HCl(842148-40-7 Free base) | Akt |
AKT Kinase Inhibitor HCl is an Akt inhibitor with antitumor activity. |